SCHEMBL4410156

SCHEMBL4410156

Cc1cc(-c2csc(NC(=O)CBr)n2)ccc1OCc1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.49
MEN1 O00255 8/20 0.48
KMT2A Q03164 8/20 0.48
TRPA1 O75762 2/20 0.46
PDE5A O76074 1/20 0.46
TRPV3 Q8NET8 1/20 0.46
TRPV4 Q9HBA0 1/20 0.46
EGFR P00533 1/20 0.45
ERBB2 P04626 1/20 0.45
CYP3A4 P08684 2/20 0.45
ROCK1 Q13464 2/20 0.45
ALDH1A1 P00352 2/20 0.44
GAA P10253 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PPARD Q03181 1/20 0.44
RAB9A P51151 2/20 0.43
POLB P06746 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13570325 0.89 MEN1 (0.52) MEN1KMT2ACYP3A4ROCK1ALDH1A1
SCHEMBL4411028 0.81 TRPA1 (0.60) MEN1KMT2ATRPA1PDE5ATRPV3
SCHEMBL13570215 0.78 TRPA1 (0.40) FFAR4MEN1KMT2ATRPA1PDE5A
SCHEMBL611935 0.75 KMT2A (0.51) MEN1KMT2ATRPA1ALDH1A1RAB9A
SCHEMBL4418963 0.75 GSTO1 (0.66) KMT2ATRPA1TRPV4ROCK1
SCHEMBL613256 0.73 KMT2A (0.48) MEN1KMT2ATRPA1ROCK1RAB9A
SCHEMBL13570207 0.73 GSTO1 (0.50) MEN1KMT2ATRPA1TRPV3TRPV4
SCHEMBL4412791 0.73 TRPA1 (0.46) KMT2ATRPA1ROCK1
SCHEMBL480701 0.72 MEN1 (0.55) MEN1KMT2ATRPA1TRPV4L3MBTL1
SCHEMBL2449783 0.71 TRPA1 (0.60) MEN1KMT2ATRPA1TRPV3TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009144548-A1 IMIDAZO [2,1-B] PURINE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2009-12-03 WO disclosed