SCHEMBL4414542

SCHEMBL4414542

O=C(NCCCO)Oc1nc2nc(Nc3ccc(F)cc3)ncc2cc1-c1ccccc1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 5/20 0.39
TBK1 Q9UHD2 7/20 0.38
PDPK1 O15530 3/20 0.36
MAPK10 P53779 2/20 0.35
MAPK9 P45984 1/20 0.35
PTK2 Q05397 2/20 0.34
CDK2 P24941 3/20 0.34
CDK9 P50750 3/20 0.34
CDC7 O00311 1/20 0.34
DAPK3 O43293 1/20 0.34
PAK4 O96013 1/20 0.34
PIM1 P11309 1/20 0.34
FLT3 P36888 1/20 0.34
GSK3B P49841 1/20 0.34
CDK5 Q00535 1/20 0.34
DYRK1A Q13627 1/20 0.34
MELK Q14680 1/20 0.34
MINK1 Q8N4C8 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
STK17A Q9UEE5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4413555 0.95 BRAF (0.38) KCNH3TBK1MAPK10MAPK9CDK2
SCHEMBL4410855 0.92 CCNT1 (0.42) TBK1PTK2CDK2CDK9CCNT1
SCHEMBL4410707 0.92 TBK1 (0.38) TBK1PDPK1MAPK10PTK2CDK2
SCHEMBL4415084 0.90 MAPK10 (0.36) TBK1MAPK10MAPK9PTK2CDK2
SCHEMBL4412920 0.90 MAPK10 (0.36) TBK1MAPK10MAPK9PTK2CDK2
SCHEMBL4411774 0.89 MAPK10 (0.36) TBK1PDPK1MAPK10MAPK9PTK2
SCHEMBL4416830 0.89 BRAF (0.44) KCNH3TBK1CDK2CDK9CCNT1
SCHEMBL4422236 0.89 CDK2 (0.33) KCNH3TBK1PDPK1MAPK10MAPK9
SCHEMBL4418433 0.89 CDK2 (0.47) MAPK10PTK2CDK2CDK9CDC7
SCHEMBL4413438 0.87 MAPK10 (0.34) TBK1MAPK10MAPK9PTK2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615921-B1 PYRIDO 2,3-D PYRIMIDIN-7-CARBOXYLIC ACID DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2009-03-18 EP claimed