SCHEMBL4418433

SCHEMBL4418433

CN(C)CCNC(=O)Oc1nc2nc(Nc3ccc(F)cc3)ncc2cc1-c1ccccc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 7/20 0.47
CCNT1 O60563 6/20 0.47
CDK9 P50750 6/20 0.47
CCNE1 P24864 3/20 0.47
CCNA2 P20248 3/20 0.43
CCNA1 P78396 2/20 0.42
BRAF P15056 1/20 0.39
IGF1R P08069 1/20 0.38
MAPK1 P28482 1/20 0.37
CDC7 O00311 1/20 0.37
CDK19 Q9BWU1 1/20 0.37
PTK2 Q05397 4/20 0.36
IKBKB O14920 1/20 0.36
CHUK O15111 1/20 0.36
IKBKG Q9Y6K9 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
MAPK10 P53779 1/20 0.35
PKM P14618 1/20 0.35
ABL1 P00519 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4410855 0.95 CCNT1 (0.42) CDK2CCNT1CDK9CCNE1CCNA2
SCHEMBL4412920 0.90 MAPK10 (0.36) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4415084 0.90 MAPK10 (0.36) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4413555 0.90 BRAF (0.38) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4416830 0.89 BRAF (0.44) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4410707 0.89 TBK1 (0.38) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4414542 0.89 KCNH3 (0.39) CDK2CCNT1CDK9CCNE1BRAF
SCHEMBL4411789 0.88 CDK2 (0.40) CDK2CCNT1CDK9CCNE1CCNA2
SCHEMBL4411774 0.88 MAPK10 (0.36) CDK2CCNT1CDK9CCNE1CDC7
SCHEMBL4417149 0.88 FGFR1 (0.39) CDK2CCNT1CDK9CCNE1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615921-B1 PYRIDO 2,3-D PYRIMIDIN-7-CARBOXYLIC ACID DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2009-03-18 EP claimed