SCHEMBL4415325

SCHEMBL4415325

COc1cc(C(=O)[C@@H]2C(=O)c3cc(-c4ccc(C(N)=O)cn4)ccc3OC23CCNCC3)cc(OC)c1-c1cnn(C)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.35
PLAU P00749 1/20 0.34
NSD2 O96028 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
FYN P06241 1/20 0.33
KCNH2 Q12809 1/20 0.32
HDAC1 Q13547 1/20 0.32
CSF1R P07333 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
TTK P33981 3/20 0.32
CCNA2 P20248 1/20 0.32
CDK2 P24941 1/20 0.32
PIK3CA P42336 1/20 0.32
ATR Q13535 1/20 0.32
MAP4K4 O95819 1/20 0.31
IGF1R P08069 2/20 0.31
FGFR1 P11362 1/20 0.31
FGFR2 P21802 1/20 0.31
FGFR3 P22607 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4430464 0.96 HSP90AA1 (0.33) HSP90AA1PLAUNSD2MKNK1MKNK2
SCHEMBL4427891 0.87 SSTR5 (0.37) KCNH2HDAC1CSF1RIRAK4MAP4K4
SCHEMBL1445071 0.82 CYP2D6 (0.33) KCNH2HDAC1
SCHEMBL4412902 0.82 ACACB (0.41) MKNK1MKNK2TTKMAP4K4IGF1R
SCHEMBL4423082 0.82 IRAK4 (0.33) KCNH2CSF1RIRAK4TTKIGF1R
SCHEMBL4412864 0.80 SSTR5 (0.34) WNT1GSK3BDYRK1A
SCHEMBL4416789 0.79 ACACB (0.38) MKNK1MKNK2CSF1RMAP4K4FGFR1
SCHEMBL4423563 0.78 TTK (0.33) TTKWNT1GSK3BDYRK1A
SCHEMBL4423456 0.78 S1PR1 (0.34) CSF1RIRAK4TTKMAP4K4WNT1
SCHEMBL4427980 0.78 GSK3B (0.33) MKNK1MKNK2CSF1RIRAK4FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP claimed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO claimed