SCHEMBL4430464

SCHEMBL4430464

CCOc1cc(C(=O)[C@@H]2C(=O)c3cc(-c4ccc(C(N)=O)cn4)ccc3OC23CCNCC3)cc(OC)c1-c1cnn(C)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.33
HDAC1 Q13547 2/20 0.32
PDE5A O76074 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
AAK1 Q2M2I8 1/20 0.32
NSD2 O96028 1/20 0.32
SSTR5 P35346 3/20 0.32
PLAU P00749 1/20 0.32
MAPK1 P28482 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
FYN P06241 1/20 0.31
KCNH2 Q12809 2/20 0.31
CYP2D6 P10635 1/20 0.31
OPRD1 P41143 1/20 0.31
CSF1R P07333 1/20 0.31
IGF1R P08069 1/20 0.30
HSD11B1 P28845 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4415325 0.96 HSP90AA1 (0.35) HSP90AA1HDAC1AAK1NSD2PLAU
SCHEMBL4427891 0.92 SSTR5 (0.37) HDAC1PDE5AHDAC2HDAC6SSTR5
SCHEMBL1445071 0.87 CYP2D6 (0.33) HDAC1PDE5AHDAC2HDAC6SSTR5
SCHEMBL4412902 0.87 ACACB (0.41) AAK1SSTR5MKNK1MKNK2IGF1R
SCHEMBL4423082 0.86 IRAK4 (0.33) AAK1KCNH2OPRD1CSF1RIGF1R
SCHEMBL4412864 0.85 SSTR5 (0.34) SSTR5
SCHEMBL4416789 0.84 ACACB (0.38) SSTR5MKNK1MKNK2CSF1RFGFR1
SCHEMBL4423456 0.83 S1PR1 (0.34) SSTR5CSF1RIRAK4
SCHEMBL4423563 0.83 TTK (0.33)
SCHEMBL4427980 0.83 GSK3B (0.33) SSTR5MKNK1MKNK2CSF1RIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed