SCHEMBL4416221

SCHEMBL4416221

CCN(C(=O)O)c1c(F)cc(N(Cc2ccccc2)Cc2ccccc2)cc1F

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
TSHR P16473 2/20 0.46
LMNA P02545 1/20 0.43
PTPN1 P18031 1/20 0.43
ALDH1A1 P00352 4/20 0.42
GLA P06280 1/20 0.42
RAB9A P51151 1/20 0.42
TSPO P30536 2/20 0.42
CYP2C19 P33261 1/20 0.41
MGLL Q99685 1/20 0.41
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
NR3C1 P04150 1/20 0.41
KDM4E B2RXH2 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2884029 0.77 CRHBP (0.53) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL14510437 0.75 TSHR (0.50) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL12346186 0.75 CYP2C19 (0.56) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL8773449 0.75 CRHBP (0.50) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL28813822 0.74 CRHBP (0.53) CRHBPCRHR2PTPN1ALDH1A1CYP2C19
SCHEMBL2887865 0.74 CRHBP (0.49) CRHBPCRHR2PTPN1ALDH1A1RAB9A
SCHEMBL3632685 0.73 CRHBP (0.46) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL3632686 0.73 CRHBP (0.46) CRHBPCRHR2TSHRPTPN1ALDH1A1
SCHEMBL8272263 0.72 NLRP3 (0.49) CRHBPCRHR2TSHRLMNAPTPN1
SCHEMBL1927316 0.72 TDP1 (0.57) TSHRALDH1A1GLARAB9ATSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742945-B1 SUBSTITUTED PHENYLAMINO-PYRIMIDINES BAYER SCHERING PHARMA AG (DE) 2009-12-30 EP disclosed
EP-1742945-A1 SUBSTITUTED PHENYLAMINO-PYRIMIDINES Bayer HealthCare AG (DE) 2007-01-17 EP disclosed
WO-2005108397-A1 SUBSTITUTED PHENYLAMINO-PYRIMIDINES BAYER HEALTHCARE AG (DE) 2005-11-17 WO disclosed