SCHEMBL4416334

SCHEMBL4416334

O=C(NCCO)Oc1nc2nc(Nc3ccc(S(=O)(=O)NCCO)cc3)ncc2cc1-c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 5/20 0.42
SYK P43405 2/20 0.42
BRAF P15056 1/20 0.38
CDK2 P24941 7/20 0.36
CDK1 P06493 4/20 0.36
CDK4 P11802 2/20 0.36
CCNE1 P24864 1/20 0.36
CCNT1 O60563 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK7 P50613 1/20 0.36
CDK9 P50750 1/20 0.36
CCNH P51946 1/20 0.36
PLK1 P53350 2/20 0.36
PLK3 Q9H4B4 2/20 0.36
PLK2 Q9NYY3 2/20 0.36
CA12 O43570 1/20 0.36
ABL1 P00519 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
KDR P35968 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4413502 0.92 CDK1 (0.36) IKBKBSYKBRAFCDK2CDK1
SCHEMBL4413555 0.88 BRAF (0.38) SYKBRAFCDK2CDK4CCNE1
SCHEMBL4412949 0.84 IKBKB (0.45) IKBKBSYKCDK2CDK1CDK4
SCHEMBL4414542 0.83 KCNH3 (0.39) BRAFCDK2CCNE1CCNT1CDK9
SCHEMBL4411774 0.82 MAPK10 (0.36) IKBKBSYKCDK2CDK1CDK4
SCHEMBL4422236 0.81 CDK2 (0.33) BRAFCDK2CDK1CDK4CCNE1
SCHEMBL4412920 0.80 MAPK10 (0.36) BRAFCDK2CDK4CCNE1CCNT1
SCHEMBL4415084 0.80 MAPK10 (0.36) BRAFCDK2CDK4CCNE1CCNT1
SCHEMBL4416830 0.79 BRAF (0.44) BRAFCDK2CCNE1CCNT1CDK9
SCHEMBL4410855 0.79 CCNT1 (0.42) BRAFCDK2CCNE1CCNT1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615921-B1 PYRIDO 2,3-D PYRIMIDIN-7-CARBOXYLIC ACID DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS HOFFMANN LA ROCHE (CH) 2009-03-18 EP claimed