SCHEMBL4417413

SCHEMBL4417413

Cc1cc2cc(C(O)(C(F)(F)F)C(F)(F)F)ccc2n1Cc1cccc(C(=O)N(C)CCN2C=CC=CC2)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.39
EPHX2 P34913 1/20 0.32
PPARG P37231 1/20 0.32
MAPK14 Q16539 1/20 0.32
BRD4 O60885 4/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
CCR2 P41597 1/20 0.31
F10 P00742 2/20 0.31
KLK1 P06870 1/20 0.31
PGR P06401 1/20 0.30
RORA P35398 1/20 0.30
RORC P51449 1/20 0.30
RORB Q92753 1/20 0.30
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1803545 0.83 MLYCD (0.58) MLYCDHDAC1HDAC2HDAC8HDAC6
SCHEMBL4414741 0.82 MAPK14 (0.42) MLYCDMAPK14BRD4HDAC1HDAC2
SCHEMBL4418588 0.81 MLYCD (0.57) MLYCDPPARGHDAC1HDAC2HDAC8
SCHEMBL1807511 0.79 MLYCD (0.42) MLYCDEPHX2PPARGMAPK14BRD4
SCHEMBL1804344 0.79 MLYCD (0.46) MLYCDPPARGNR1H2NR1H3
SCHEMBL1811315 0.77 CCR2 (0.51) BRD4HDAC1HDAC2HDAC8HDAC6
SCHEMBL4420743 0.77 HSD11B1 (0.45) MLYCDEPHX2PPARGRORARORC
SCHEMBL4421334 0.77 CDK4 (0.55) MLYCD
SCHEMBL4415610 0.77 MLYCD (0.44) MLYCDPPARGBRD4HDAC1HDAC2
SCHEMBL1813000 0.75 F10 (0.48) BRD4HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756096-B1 INDOLYL DERIVATIVES AS LIVER-X-RECEPTOR MODULATORS HOFFMANN LA ROCHE (CH) 2009-08-12 EP claimed