SCHEMBL4417585

SCHEMBL4417585

CNc1nc(N[C@H]2CCN(C3(CS(=O)(=O)c4ccccc4)CCC(NCC(C)C)CC3)C2=O)c2cc(Cl)ccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.40
NSD2 O96028 1/20 0.38
CNR2 P34972 1/20 0.35
HTR3A P46098 1/20 0.35
PDE5A O76074 6/20 0.34
F10 P00742 1/20 0.34
CCR2 P41597 1/20 0.34
CCR5 P51681 1/20 0.34
CAMK2D Q13557 1/20 0.34
KMT2A Q03164 1/20 0.34
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33
NTRK1 P04629 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4416711 0.92 CNR1 (0.37) CNR1CNR2PDE5AF10CCR2
SCHEMBL4413722 0.92 F10 (0.35) CNR1CNR2F10CCR2CCR5
SCHEMBL4421724 0.91 F10 (0.36) CNR1F10CCR2CCR5KMT2A
SCHEMBL4428598 0.91 F10 (0.36) CNR1CNR2F10CCR2CCR5
SCHEMBL4415059 0.90 CCR2 (0.35) CNR1CNR2F10CCR2CCR5
SCHEMBL4420896 0.90 CCR2 (0.36) CNR1NSD2CNR2F10CCR2
SCHEMBL4417993 0.90 NSD2 (0.39) CNR1NSD2F10CCR2CCR5
SCHEMBL4427802 0.90 F10 (0.34) CNR1CNR2F10CCR2CCR5
SCHEMBL5029465 0.89 CCR2 (0.43) CNR1NSD2CNR2HTR3APDE5A
SCHEMBL4426067 0.84 CNR1 (0.40) CNR1NSD2CNR2CCR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606255-B1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2009-11-11 EP claimed