SCHEMBL4418059

SCHEMBL4418059

O=C(O)CNC(=O)c1nc(Cl)c2cccc(I)c2c1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 14/20 0.57
FTO Q9C0B1 4/20 0.57
BBOX1 O75936 2/20 0.57
KDM5B Q9UGL1 2/20 0.45
KDM2A Q9Y2K7 2/20 0.45
THRA P10827 1/20 0.45
THRB P10828 1/20 0.45
KDM6B O15054 2/20 0.43
EGLN3 Q9H6Z9 2/20 0.42
TET3 O43151 1/20 0.42
VEGFA P15692 1/20 0.42
FLT1 P17948 1/20 0.42
ASPH Q12797 1/20 0.42
TET2 Q6N021 1/20 0.42
KDM8 Q8N371 1/20 0.42
OGFOD1 Q8N543 1/20 0.42
TET1 Q8NFU7 1/20 0.42
HIF1AN Q9NWT6 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5027666 0.84 EGLN1 (0.68) EGLN1FTOBBOX1THRATHRB
SCHEMBL522656 0.84 EGLN1 (0.71) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL4757084 0.82 EGLN1 (0.61) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL4419152 0.81 EGLN1 (0.53) EGLN1FTOBBOX1THRATHRB
SCHEMBL4755920 0.79 EGLN1 (0.51) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL523235 0.79 EGLN1 (0.70) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL5325511 0.75 EGLN1 (0.61) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL5315453 0.75 EGLN1 (0.61) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL522478 0.74 EGLN1 (0.56) EGLN1FTOBBOX1KDM5BKDM2A
SCHEMBL4757876 0.74 EGLN1 (0.59) EGLN1FTOBBOX1KDM5BKDM2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008040002-A9 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR HIF MODULATING COMPOUNDS HUTCHINSON FRED CANCER RES (US) 2009-04-16 WO disclosed
WO-2009002533-A1 INFLAMMATORY BOWEL DISEASE THERAPIES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2008-12-31 WO disclosed
WO-2008040002-A2 METHODS, COMPOSITIONS AND ARTICLES OF MANUFACTURE FOR HIF MODULATING COMPOUNDS FRED HUTCHINSON CANCER RESEARCH CENTER (US) 2008-04-03 WO disclosed