SCHEMBL4419617

SCHEMBL4419617

Fc1cc(Br)cc(OCc2ccccc2)c1F.O=C(O)Cc1cc(F)c(F)c(OCc2ccccc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.52
PTGER1 P34995 3/20 0.44
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
PTPN1 P18031 2/20 0.43
NPC1 O15118 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
PTGER4 P35408 1/20 0.42
PTGER3 P43115 1/20 0.42
PTGER2 P43116 1/20 0.42
LRRK2 Q5S007 1/20 0.42
S1PR5 Q9H228 1/20 0.41
SLC26A3 P40879 1/20 0.41
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
FOLH1 Q04609 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
FFAR1 O14842 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3799950 0.92 RXRB (0.49) PTGER1RXRARXRBRXRGPTPN1
SCHEMBL3795791 0.87 KDM1A (0.64) KDM1APTGER1NPC1MRGPRX4LRRK2
SCHEMBL3954112 0.77 S1PR5 (0.60) PTGER1RXRARXRBRXRGNPC1
SCHEMBL29510818 0.77 S1PR5 (0.60) PTGER1RXRARXRBRXRGNPC1
SCHEMBL13014915 0.77 THRA (0.52) KDM1APTGER1RXRARXRBRXRG
SCHEMBL5527936 0.76 PKM (0.53) PTPN1
SCHEMBL24277672 0.75 PTPN1 (0.56) PTGER1RXRARXRBRXRGPTPN1
SCHEMBL17893533 0.75 KDM1A (0.51) KDM1APTGER1
SCHEMBL28759062 0.75 FFAR1 (0.51) KDM1APTGER1RXRARXRBRXRG
SCHEMBL25337360 0.74 MRGPRX4 (0.59) PTGER1NPC1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120898-A1 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2009-11-25 EP disclosed
WO-2008077009-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-06-26 WO disclosed