SCHEMBL4421333

SCHEMBL4421333

Cc1ccc(-c2ncc(C(=O)O)cc2Cl)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH5 P11766 1/20 0.44
PTGS2 P35354 6/20 0.44
PTGS1 P23219 2/20 0.44
ABCC4 O15439 1/20 0.44
ABCB11 O95342 1/20 0.44
PDE4D Q08499 1/20 0.44
MAPK14 Q16539 1/20 0.44
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NAPRT Q6XQN6 1/20 0.40
KMO O15229 2/20 0.39
GRM5 P41594 1/20 0.39
MAP4K4 O95819 3/20 0.39
TSHR P16473 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.38
SLC22A12 Q96S37 1/20 0.38
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138792 0.85 PTGS2 (0.41) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL4413866 0.80 ADH5 (0.43) ADH5PTGS2NAPRTKMOMAP4K4
SCHEMBL14422878 0.78 PTGS2 (0.65) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL4181890 0.78 PTGS2 (0.57) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL1543442 0.75 HPGDS (0.48) ADH5KMO
SCHEMBL29788311 0.74 MKNK1 (0.58) HDAC1HDAC6MAP4K4TSHRALDH1A1
SCHEMBL2038607 0.74 MKNK1 (0.58) HDAC1HDAC6MAP4K4TSHRALDH1A1
SCHEMBL3628259 0.73 GRM5 (0.67) GRM5NPSR1
SCHEMBL181465 0.73 HDAC1 (0.62) HDAC1HDAC6NAPRTALDH1A1
SCHEMBL30544993 0.73 HDAC1 (0.62) HDAC1HDAC6NAPRTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054405-B1 NOVEL BIARYL BENZOIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAE WOONG PHARMA (KR) 2013-09-18 EP disclosed
EP-2054405-A1 NOVEL BIARYL BENZOIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2009-05-06 EP disclosed
WO-2008007900-A1 NOVEL BIARYL BENZOIMIDAZOLE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2008-01-17 WO disclosed