SCHEMBL4421630

SCHEMBL4421630

O=C1OCCN1CC(=O)N(Cc1ccsc1)C1CCN(C2CNC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 10/20 0.52
NAAA Q02083 1/20 0.38
KCNH2 Q12809 4/20 0.35
AGTR2 P50052 2/20 0.34
SIGMAR1 Q99720 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
OPRM1 P35372 4/20 0.33
OPRD1 P41143 4/20 0.33
OPRK1 P41145 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4551472 0.81 CCR5 (0.49) CCR5NAAAKCNH2SIGMAR1NPC1
SCHEMBL4415713 0.75 CCR5 (0.57) CCR5KCNH2
SCHEMBL4416636 0.75 CCR5 (0.52) CCR5KCNH2AGTR2
SCHEMBL3761943 0.70 CCR5 (0.91) CCR5KCNH2
SCHEMBL3761945 0.70 CCR5 (0.91) CCR5KCNH2
SCHEMBL3752682 0.70 CCR5 (0.85) CCR5KCNH2
SCHEMBL3752686 0.70 CCR5 (0.85) CCR5KCNH2
SCHEMBL3756667 0.70 CCR5 (1.00) CCR5KCNH2
SCHEMBL3756671 0.70 CCR5 (1.00) CCR5KCNH2
SCHEMBL13052008 0.69 CCR5 (0.77) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088860-A1 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2009-08-19 EP disclosed
WO-2008070758-A1 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2008-06-12 WO disclosed