Bicarbonate

Bicarbonate

SCHEMBL4423929

COc1cccc(Cl)c1CC(=O)NC1CCCCC1C.O=C(O)O

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 9/20 0.54
TAS1R1 Q7RTX1 9/20 0.54
TAS1R2 Q8TE23 5/20 0.54
LMNA P02545 3/20 0.49
KMT2A Q03164 2/20 0.49
HPGD P15428 1/20 0.49
ATM Q13315 1/20 0.49
TSHR P16473 1/20 0.47
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HTT P42858 1/20 0.47
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7620719 0.89 TAS1R3 (0.63) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4423930 0.86 KMT2A (0.62) KMT2AHPGDATMTSHRKDM4E
Bicarbonate SCHEMBL4431556 0.85 KMT2A (0.60) KMT2AHPGDATMALDH1A1HTT
Bicarbonate SCHEMBL4422720 0.85 KMT2A (0.60) KMT2AHPGDATMALDH1A1HTT
Bicarbonate SCHEMBL7620822 0.84 ALDH1A1 (0.58) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4426525 0.81 KMT2A (0.63) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4435106 0.81 KMT2A (0.55) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4428857 0.80 KMT2A (0.51) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4435414 0.78 KMT2A (0.61) TAS1R3TAS1R1TAS1R2LMNAKMT2A
Bicarbonate SCHEMBL4423951 0.77 KMT2A (0.60) TAS1R3TAS1R1TAS1R2LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741700-B1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2009-10-07 EP disclosed
EP-0741700-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AG (DE) 1996-11-13 EP disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed