Bicarbonate

Bicarbonate

SCHEMBL4428857

COc1cccc(Cl)c1CC(=O)NC1CCCC(C)C1.O=C(O)O

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
GAA P10253 1/20 0.46
SIGMAR1 Q99720 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 1/20 0.44
MTNR1A P48039 2/20 0.42
MTNR1B P49286 2/20 0.42
CXCR6 O00574 2/20 0.42
ATM Q13315 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
MEN1 O00255 2/20 0.41
RAB9A P51151 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7622727 0.90 KMT2A (0.63) KMT2ASIGMAR1ALDH1A1ATMMEN1
Bicarbonate SCHEMBL4423930 0.89 KMT2A (0.62) KMT2AGAASIGMAR1L3MBTL1ALDH1A1
Bicarbonate SCHEMBL4422720 0.88 KMT2A (0.60) KMT2ASIGMAR1L3MBTL1ALDH1A1HPGD
Bicarbonate SCHEMBL4431556 0.88 KMT2A (0.60) KMT2ASIGMAR1L3MBTL1ALDH1A1HPGD
Bicarbonate SCHEMBL4426525 0.86 KMT2A (0.63) KMT2AGAASIGMAR1L3MBTL1ALDH1A1
Bicarbonate SCHEMBL4435106 0.86 KMT2A (0.55) KMT2AGAASIGMAR1L3MBTL1ALDH1A1
Bicarbonate SCHEMBL7614611 0.84 ALDH1A1 (0.61) KMT2AGAASIGMAR1ALDH1A1MAPT
Bicarbonate SCHEMBL4435414 0.81 KMT2A (0.61) KMT2AGAASIGMAR1L3MBTL1ALDH1A1
Bicarbonate SCHEMBL4423929 0.80 TAS1R3 (0.54) KMT2AALDH1A1HPGDATMTAS1R3
Bicarbonate SCHEMBL4423951 0.80 KMT2A (0.60) KMT2AGAASIGMAR1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741700-B1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2009-10-07 EP disclosed
EP-0741700-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AG (DE) 1996-11-13 EP disclosed
WO-1995020572-A1 1-H-3-ARYLPYRROLIDINE-2,4-DIONE DERIVATIVES AS PEST-CONTROL AGENTS BAYER AKTIENGESELLSCHAFT (DE) 1995-08-03 WO disclosed