Dichloroacetic Acid

Dichloroacetic Acid

SCHEMBL4424191

O=C(O)C(Cl)Cl.c1cc2ccc1o2

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PDK1PDK2PDK3PDK4

The experimentally established mechanism targets of Dichloroacetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.53
ALDH1A1 P00352 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP2D6 P10635 1/20 0.33
SRC P12931 1/20 0.33
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
PTPN1 P18031 1/20 0.32
PTPN7 P35236 1/20 0.32
BLM P54132 1/20 0.32
ESR2 Q92731 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 2/20 0.31
PDPK1 O15530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5273126 0.82 LMNA (0.35) LMNAALDH1A1KMT2AMEN1MAPT
SCHEMBL5334623 0.79 ALDH1A1 (0.36) LMNAALDH1A1KMT2AMEN1MAPT
Acetic Acid SCHEMBL11212519 0.75 FFAR3 (0.44) ALDH1A1KMT2AMEN1MAPTHPGD
Dichloroacetic Acid SCHEMBL7496768 0.75 LMNA (0.62) LMNAALDH1A1KMT2AMEN1MAPT
Dichloroacetic Acid SCHEMBL11843218 0.75 LMNA (0.62) LMNAALDH1A1KMT2AMEN1MAPT
Chloroacetic Acid SCHEMBL11683671 0.74 TSHR (0.53) LMNAALDH1A1KMT2AMEN1MAPT
SCHEMBL27587735 0.74 ALDH1A1 (0.30) ALDH1A1
Dichloroacetic Acid SCHEMBL28158662 0.73 LMNA (0.83) LMNAALDH1A1KMT2AMEN1MAPT
Dichloroacetic Acid SCHEMBL5307050 0.72 LMNA (1.00) LMNAALDH1A1KMT2AMEN1MAPT
Dichloroacetic Acid SCHEMBL7777 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1855527-A4 LIMONENE-CONTAINING HERBICIDE COMPOSITIONS, HERBICIDE CONCENTRATE FORMULATIONS AND METHODS FOR MAKING AND USING SAME CUTTING EDGE FORMULATIONS INC (US) 2009-06-10 EP disclosed
EP-1855527-A2 LIMONENE-CONTAINING HERBICIDE COMPOSITIONS, HERBICIDE CONCENTRATE FORMULATIONS AND METHODS FOR MAKING AND USING SAME Cutting Edge Formulations, Inc. (US) 2007-11-21 EP disclosed
WO-2006094126-A2 LIMONENE-CONTAINING HERBICIDE COMPOSITIONS, HERBICIDE CONCENTRATE FORMULATIONS AND METHODS FOR MAKING AND USING SAME CUTTING EDGE FORMULATIONS, INC. (US) 2006-09-08 WO disclosed
EP-1051496-A1 WHISKER-MEDIATED TRANSFORMATION OF PLANT CELL AGGREGATES AND PLANT TISSUES AND REGENERATION OF PLANTS THEREOF Dow Agrosciences LLC (US) 2000-11-15 EP disclosed
WO-1999038979-A1 WHISKER-MEDIATED TRANSFORMATION OF PLANT CELL AGGREGATES AND PLANT TISSUES AND REGENERATION OF PLANTS THEREOF DOW AGROSCIENCES LLC (US) 1999-08-05 WO disclosed
WO-1998050569-A2 NUCLEOTIDE SEQUENCES OF MAIZE OLEOYL-ACP THIOESTERASE AND PALMITOYL-ACP THIOESTERASE GENES AND THEIR USE IN THE MODIFICATION OF FATTY ACID CONTENT OF OIL DOW AGROSCIENCES LLC (US) 1998-11-12 WO disclosed
US-4013706-A FROM A CYANAMIDE; ACID CATALYST SUCRERIES DU SOISSONNAIS ET COMPAGNIE SUCRIERE (FR) 1977-03-22 US disclosed