SCHEMBL5423936

SCHEMBL5423936

CCOC(=O)c1cc(C#N)c(N2CCNC(CCC(=O)OC(C)(C)C)C2)nc1C(F)(F)CF

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
P2RY12 Q9H244 16/20 0.46
KDM4E B2RXH2 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ACACB O00763 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930058 0.93 ALDH1A1 (0.65) ALDH1A1P2RY12KDM4ENPSR1ACACB
SCHEMBL5423937 0.87 ALDH1A1 (0.51) ALDH1A1P2RY12KDM4ENPSR1ACACB
SCHEMBL4425609 0.81 ALDH1A1 (0.84) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL4104450 0.74 P2RY12 (0.68) ALDH1A1P2RY12
SCHEMBL3926740 0.73 ALDH1A1 (1.00) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL30999844 0.73 ALDH1A1 (1.00) ALDH1A1P2RY12KDM4ENPSR1
SCHEMBL4117402 0.72 P2RY12 (0.69) ALDH1A1P2RY12
SCHEMBL4094945 0.72 P2RY12 (0.68) P2RY12
SCHEMBL4105670 0.72 P2RY12 (0.46) P2RY12
SCHEMBL4097642 0.70 P2RY12 (0.86) P2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836189-A1 NOVEL PYRIDINE COMPOUNDS AstraZeneca AB (SE) 2007-09-26 EP disclosed
WO-2006073361-A1 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2006-07-13 WO disclosed