SCHEMBL4430723

SCHEMBL4430723

Cc1c[nH]c(=O)c(Cc2ccccc2)c1CC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.42
AKR1B1 P15121 1/20 0.42
ALDH1A1 P00352 4/20 0.41
PTGDR2 Q9Y5Y4 3/20 0.41
KDM4E B2RXH2 4/20 0.40
GAA P10253 2/20 0.40
MAPT P10636 2/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
KAT8 Q9H7Z6 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
DAO P14920 1/20 0.38
TYMP P19971 1/20 0.38
PIM1 P11309 1/20 0.38
LMNA P02545 1/20 0.38
NQO1 P15559 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4431452 0.85 HSD17B10 (0.47) ALDH1A1KDM4EGAAKMT2ASMN1; SMN2
SCHEMBL9356524 0.73 KDM4E (0.47) IDH1ALDH1A1KDM4EGAAMAPT
SCHEMBL7378429 0.71 KDM4E (0.48) AKR1B1ALDH1A1PTGDR2KDM4EGAA
SCHEMBL1346299 0.71 IDH1 (0.49) IDH1ALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL5396566 0.70 NOTUM (0.50) AKR1B1ALDH1A1KDM4EGAAMAPT
Hydrochloric Acid SCHEMBL9356148 0.70 ALDH1A1 (0.40) IDH1ALDH1A1KDM4EMAPTMEN1
SCHEMBL18937921 0.69 AKR1B1 (0.47) IDH1AKR1B1ALDH1A1PTGDR2KDM4E
SCHEMBL5199231 0.68 ALDH1A1 (0.47) ALDH1A1KDM4EGAAMAPTMEN1
SCHEMBL18937923 0.68 AKR1B1 (0.42) IDH1AKR1B1ALDH1A1PTGDR2KDM4E
Phenylacetic Acid SCHEMBL28136536 0.66 AKR1B1 (0.77) AKR1B1ALDH1A1GAASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed