SCHEMBL4431041

SCHEMBL4431041

CC(=O)NCc1ccncc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 14/20 0.46
KDM6B O15054 6/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 3/20 0.43
KDM4A O75164 3/20 0.43
KDM4D Q6B0I6 3/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MTNR1A P48039 1/20 0.42
USP2 O75604 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP11B2 P19099 1/20 0.40
KDM5C P41229 1/20 0.40
SLCO1B1 Q9Y6L6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10061709 0.80 ALDH1A1 (0.45) KDM4EALDH1A1MAPTTDP1MTNR1A
Acetic Acid SCHEMBL16666943 0.80 KDM4C (0.49) KDM4CKDM6BKMT2AKDM4EKDM4A
SCHEMBL30465694 0.79 KDM4C (0.51) KDM4CKDM6BKMT2AKDM4EKDM4A
SCHEMBL123203 0.79 KDM4C (0.51) KDM4CKDM6BKMT2AKDM4EKDM4A
SCHEMBL16196603 0.79 KMT2A (0.48) KMT2AL3MBTL1MTNR1ANPSR1CYP11B2
SCHEMBL2370442 0.78 KDM4C (0.46) KDM4CKDM6BKMT2AKDM4EKDM4A
SCHEMBL14960629 0.77 SOST (0.54) KDM4CALDH1A1TDP1MTNR1ANPSR1
SCHEMBL9848860 0.76 HTT (0.57) KMT2AKDM4EALDH1A1L3MBTL1MTNR1A
SCHEMBL3880004 0.75 KDM4C (0.50) KDM4CKDM6BKMT2AKDM4EKDM4A
SCHEMBL258369 0.75 KDM4C (0.51) KDM4CKDM6BKMT2AKDM4EKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124913-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS Novartis AG (CH) 2009-12-02 EP disclosed
WO-2008077597-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS NOVARTIS AG (CH) 2008-07-03 WO disclosed