SCHEMBL4432784

SCHEMBL4432784

CNC(=O)[C@@H](NCCC(c1ccc(C)cc1)c1ccc(F)c(C)c1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.51
CNR2 P34972 2/20 0.51
CASR P41180 2/20 0.47
ALDH1A1 P00352 7/20 0.42
KDM4E B2RXH2 2/20 0.42
KMT2A Q03164 1/20 0.41
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MAPT P10636 2/20 0.39
ALOX12 P18054 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CHRM2 P08172 1/20 0.39
HTR1A P08908 1/20 0.39
ADRA2A P08913 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
CHRM1 P11229 1/20 0.39
SMPD1 P17405 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434615 1.00 CNR1 (0.51) CNR1CNR2CASRALDH1A1KDM4E
SCHEMBL4433690 1.00 CNR1 (0.51) CNR1CNR2CASRALDH1A1KDM4E
SCHEMBL4429219 1.00 CNR1 (0.51) CNR1CNR2CASRALDH1A1KDM4E
SCHEMBL4433145 0.96 CNR1 (0.45) CNR1CNR2CASRALDH1A1KDM4E
SCHEMBL4430647 0.89 KDM4E (0.46) CNR1CNR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4441795 0.89 KDM4E (0.46) CNR1CNR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4435883 0.88 EPHX2 (0.47) CNR1CNR2ALDH1A1KDM4ELMNA
SCHEMBL4430907 0.88 ALDH1A1 (0.41) CNR1CNR2ALDH1A1KDM4EKMT2A
SCHEMBL4441392 0.88 ALDH1A1 (0.41) CNR1CNR2ALDH1A1KDM4EKMT2A
SCHEMBL4432435 0.87 CNR1 (0.49) CNR1CNR2CASRALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed