SCHEMBL4435883

SCHEMBL4435883

CNC(=O)[C@H](NCC[C@@H](c1ccc(S(C)(=O)=O)cc1)c1ccc(F)c(C)c1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 10/20 0.47
LMNA P02545 1/20 0.43
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYP2J2 P51589 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434615 0.88 CNR1 (0.51) LMNAALDH1A1CNR1CNR2KDM4E
SCHEMBL4432784 0.88 CNR1 (0.51) LMNAALDH1A1CNR1CNR2KDM4E
SCHEMBL4429219 0.88 CNR1 (0.51) LMNAALDH1A1CNR1CNR2KDM4E
SCHEMBL4433690 0.88 CNR1 (0.51) LMNAALDH1A1CNR1CNR2KDM4E
SCHEMBL4433145 0.85 CNR1 (0.45) LMNAALDH1A1CNR1CNR2KDM4E
SCHEMBL4441795 0.84 KDM4E (0.46) EPHX2ALDH1A1CNR1CNR2KDM4E
SCHEMBL4430647 0.84 KDM4E (0.46) EPHX2ALDH1A1CNR1CNR2KDM4E
SCHEMBL4441392 0.83 ALDH1A1 (0.41) ALDH1A1CNR1CNR2KDM4E
SCHEMBL4430907 0.83 ALDH1A1 (0.41) ALDH1A1CNR1CNR2KDM4E
SCHEMBL4436024 0.82 P2RX7 (0.44) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed