SCHEMBL4433145

SCHEMBL4433145

CNC(=O)[C@@H](NCC[C@@H](c1ccc(C)cc1)c1ccc(F)c(C)c1)c1ccc(C)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
CASR P41180 1/20 0.41
SLC6A3 Q01959 3/20 0.40
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433690 0.96 CNR1 (0.51) CNR1CNR2CASRSLC6A3HTR1A
SCHEMBL4432784 0.96 CNR1 (0.51) CNR1CNR2CASRSLC6A3HTR1A
SCHEMBL4434615 0.96 CNR1 (0.51) CNR1CNR2CASRSLC6A3HTR1A
SCHEMBL4429219 0.96 CNR1 (0.51) CNR1CNR2CASRSLC6A3HTR1A
SCHEMBL4434471 0.86 CNR1 (0.43) CNR1CNR2CASRSLC6A3HTR1A
SCHEMBL4441783 0.86 P2RX7 (0.38) CNR1CNR2
SCHEMBL4435812 0.86 P2RX7 (0.38) CNR1CNR2
SCHEMBL4441795 0.86 KDM4E (0.46) CNR1CNR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4430647 0.86 KDM4E (0.46) CNR1CNR2ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4435883 0.85 EPHX2 (0.47) CNR1CNR2ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed