SCHEMBL4433024

SCHEMBL4433024

CNC(=O)C(NCCC(c1ccc(C(F)(F)F)cc1)c1cc(C)ccc1F)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
CCR2 P41597 8/20 0.43
ALDH1A1 P00352 2/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
TACR1 P25103 2/20 0.39
TACR3 P29371 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ULK1 O75385 1/20 0.39
HDAC4 P56524 1/20 0.38
ALOX5 P09917 1/20 0.38
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441220 1.00 KDM4E (0.43) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4429663 0.94 CCR2 (0.43) KDM4ECCR2ALDH1A1CTDSP1TACR1
SCHEMBL4440273 0.89 KDM4E (0.45) KDM4ECCR2ALDH1A1CTDSP1TACR1
SCHEMBL4438661 0.89 KDM4E (0.45) KDM4ECCR2ALDH1A1CTDSP1TACR1
SCHEMBL4427927 0.89 CNR1 (0.51) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4434552 0.89 CNR1 (0.51) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4428071 0.87 KDM4E (0.48) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4441795 0.87 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4430286 0.87 KDM4E (0.48) KDM4ECCR2ALDH1A1CTDSP1CNR1
SCHEMBL4430647 0.87 KDM4E (0.46) KDM4ECCR2ALDH1A1CTDSP1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed