SCHEMBL4433057

SCHEMBL4433057

CNc1ccc(-c2ccccc2Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.58
MAOB P27338 2/20 0.47
DHODH Q02127 1/20 0.47
TSHR P16473 1/20 0.46
USP7 Q93009 1/20 0.41
GFER P55789 1/20 0.41
MAT2A P31153 1/20 0.40
KCNH2 Q12809 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KIF11 P52732 1/20 0.39
MEN1 O00255 1/20 0.39
APP P05067 1/20 0.39
GLA P06280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5141361 0.84 TSHR (0.57) TSHRGFERCYP3A4HSD17B10KIF11
SCHEMBL25973862 0.80 TSHR (0.59) CYP2A6TSHRGFERMAPK1HSD17B10
SCHEMBL28788627 0.79 CYP2A6 (0.52) CYP2A6MAOBDHODHUSP7HSD17B10
SCHEMBL22270544 0.78 DPP4 (0.44) CYP1A2CYP3A4CYP2D6CYP2C9MAPK1
SCHEMBL6674385 0.77 CA12 (0.48) TSHRGFERCYP1A2CYP3A4CYP2D6
SCHEMBL27636093 0.76 CSNK2A1 (0.49) CYP2A6DHODHTSHRHSD17B10HSD11B1
SCHEMBL27717693 0.76 CYP2A6 (0.48) CYP2A6MAOBDHODHUSP7TAAR1
SCHEMBL1045000 0.76 CYP2A6 (0.65) CYP2A6MAOBTSHRUSP7TDP1
SCHEMBL23546571 0.75 TSHR (0.46) TSHRGFERCYP3A4HSD17B10KIF11
SCHEMBL6490058 0.75 ALDH1A1 (0.58) TSHRGFERMAPK1KIF11MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009057133-A2 A PROCESS FOR THE SYNTHESIS OF 2-[2-[4-[(4-CHLOROPHENYL)PHENYL METHYL]-1-PIPERAZINYL] ETHOXY ACETIC ACID GLENMARK GENERICS LIMITED (IN) 2009-05-07 WO disclosed
CN-1708476-A Novel amide compounds having MCH-antagonistic action and medicaments comprising these compounds BOEHRINGER INGELHEIM PHARMA (DE) 2005-12-14 CN disclosed