SCHEMBL5161949

SCHEMBL5161949

NCCC(c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.67
SLC6A2 P23975 4/20 0.62
SLC6A4 P31645 4/20 0.62
SLC6A3 Q01959 4/20 0.62
KCNK2 O95069 2/20 0.62
KCNH2 Q12809 2/20 0.62
CACNA1C Q13936 2/20 0.62
SLC7A5 Q01650 4/20 0.54
HTR2A P28223 2/20 0.52
ACP3 P15309 1/20 0.49
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
LMNA P02545 4/20 0.47
NPC1 O15118 2/20 0.47
CYP2D6 P10635 2/20 0.47
CYP2C19 P33261 2/20 0.47
MTOR P42345 2/20 0.47
RAB9A P51151 2/20 0.47
TSHR P16473 2/20 0.47
CYP3A4 P08684 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4433367 0.98 HRH1 (0.64) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL23960430 0.87 CYP19A1 (0.54) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL4432789 0.86 SLC6A2 (0.48) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL605443 0.85 HTR2A (0.64) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
Hydrochloric Acid SCHEMBL4430219 0.84 SLC6A2 (0.47) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL4433142 0.82 SLC6A2 (0.55) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL158098 0.82 HRH1 (1.00) HRH1SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL7294209 0.81 HRH3 (0.48) HRH1SLC6A2SLC6A4SLC6A3KCNK2
SCHEMBL4432893 0.81 SLC6A2 (0.51) HRH1SLC6A2SLC6A4SLC6A3KCNK2
Hydrochloric Acid SCHEMBL4441383 0.80 SLC6A2 (0.54) HRH1SLC6A2SLC6A4SLC6A3KCNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748982-A1 (4, 5, 6, 7-TETRAHYDRO-1-H-INDOL-7-YL) ACETIC ACID DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME LTD. (GB) 2007-02-07 EP disclosed
WO-2005108362-A1 (4, 5, 6, 7-TETRAHYDRO-1-H-INDOL-7-YL) ACETIC ACID DERIVATIVES FOR TREATMENT OF ALZHEIMER'S DISEASE MERCK SHARP & DOHME LIMITED (GB) 2005-11-17 WO disclosed