SCHEMBL4432789

SCHEMBL4432789

Cc1ccc(C(CCN)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.48
SLC6A4 P31645 2/20 0.48
SLC6A3 Q01959 2/20 0.48
KCNK2 O95069 1/20 0.48
KCNH2 Q12809 1/20 0.48
CACNA1C Q13936 1/20 0.48
HRH1 P35367 1/20 0.47
CYP19A1 P11511 2/20 0.43
TAAR1 Q96RJ0 1/20 0.43
SLC7A5 Q01650 4/20 0.41
UTS2R Q9UKP6 2/20 0.40
KIF11 P52732 3/20 0.40
GRM8 O00222 1/20 0.40
GRM4 Q14833 1/20 0.40
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5161949 0.86 HRH1 (0.67) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL13930329 0.85 HRH1 (0.62) SLC6A2SLC6A4SLC6A3KCNH2HRH1
Hydrochloric Acid SCHEMBL4433367 0.84 HRH1 (0.64) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL23960430 0.84 CYP19A1 (0.54) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL4433142 0.82 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
Hydrochloric Acid SCHEMBL4430219 0.81 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
Hydrochloric Acid SCHEMBL4441383 0.81 SLC6A2 (0.54) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL27790948 0.79 BCHE (0.40) CYP19A1UTS2RKIF11
SCHEMBL4434677 0.77 CASR (0.45) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL12569047 0.76 BCHE (0.42) TAAR1UTS2RKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed