SCHEMBL4433334

SCHEMBL4433334

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1ccccc1F

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 13/20 0.52
HDAC3 O15379 2/20 0.52
HDAC7 Q8WUI4 2/20 0.52
HDAC8 Q9BY41 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HDAC9 Q9UKV0 2/20 0.52
HDAC5 Q9UQL6 2/20 0.52
NCOR2 Q9Y618 2/20 0.52
HDAC1 Q13547 1/20 0.52
EEF2K O00418 1/20 0.44
ACP3 P15309 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CNR2 P34972 1/20 0.40
TACR1 P25103 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4436009 0.85 MEN1 (0.43) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL22917200 0.84 GAA (0.50) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL4433967 0.84 ACP3 (0.41) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL28226380 0.83 HDAC4 (0.46) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL4432350 0.82 AKR1C3 (0.45) ACP3AKR1C3AKR1C2CES2CES1
SCHEMBL2304585 0.82 ACP3 (0.56) EEF2KACP3CES2CES1CNR2
SCHEMBL2304513 0.81 CNR2 (0.47) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL4428068 0.81 AKR1C3 (0.41) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL22917054 0.80 CES2 (0.48) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL27792689 0.78 HDAC4 (0.42) HDAC4HDAC3HDAC7HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed