SCHEMBL4436009

SCHEMBL4436009

CC(=O)C(c1ccc(C(F)(F)F)cc1)c1ccccc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
CNR2 P34972 1/20 0.43
ACP3 P15309 1/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
CTSA P10619 1/20 0.40
TACR1 P25103 3/20 0.40
ALDH1A1 P00352 1/20 0.38
HDAC4 P56524 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4433334 0.85 HDAC4 (0.52) CNR2ACP3CES2CES1TACR1
SCHEMBL4433967 0.84 ACP3 (0.41) CNR2ACP3CES2CES1CTSA
SCHEMBL4432350 0.82 AKR1C3 (0.45) HTTACP3CES2CES1TACR1
SCHEMBL2304585 0.82 ACP3 (0.56) RAB9ACNR2ACP3CES2CES1
SCHEMBL12780403 0.82 ACP3 (0.51) MEN1KMT2AACP3ALDH1A1HDAC4
SCHEMBL28227221 0.81 ALDH1A1 (0.44) KMT2ACNR2ACP3ALDH1A1
SCHEMBL22917035 0.78 ESR1 (0.46) MEN1MAPTRAB9AKMT2AACP3
SCHEMBL4432335 0.77 CES2 (0.41) MAPTACP3CES2CES1TACR1
SCHEMBL4428068 0.75 AKR1C3 (0.41) CES2CES1HDAC4HDAC3HDAC1
SCHEMBL4434012 0.75 TRPM8 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed