SCHEMBL2304585

SCHEMBL2304585

CC(=O)C(c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 1/20 0.56
TACR1 P25103 7/20 0.51
PTPN1 P18031 1/20 0.49
PDPK1 O15530 1/20 0.48
CNR2 P34972 1/20 0.48
CES2 O00748 1/20 0.46
CES1 P23141 1/20 0.46
HSD11B1 P28845 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
NR4A1 P22736 1/20 0.45
NR4A2 P43354 1/20 0.45
NR4A3 Q92570 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CACNA1A O00555 1/20 0.45
CACNA2D1 P54289 1/20 0.45
CACNA1B Q00975 1/20 0.45
CACNB1 Q02641 1/20 0.45
CACNA1C Q13936 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438527 0.87 CES2 (0.50) ACP3TACR1CES2CES1ALDH1A1
SCHEMBL27683652 0.85 ACP3 (0.59) ACP3TACR1PTPN1PDPK1CNR2
SCHEMBL11103452 0.85 ACP3 (0.55) ACP3TACR1CES2ALDH1A1RAB9A
SCHEMBL396389 0.82 L3MBTL1 (0.56) CES2CES1ALDH1A1
Benzene SCHEMBL27414119 0.82 L3MBTL1 (0.56) CES2CES1ALDH1A1
SCHEMBL4436009 0.82 MEN1 (0.43) ACP3TACR1PTPN1CNR2CES2
SCHEMBL4433334 0.82 HDAC4 (0.52) ACP3TACR1CNR2CES2CES1
SCHEMBL28212173 0.82 ACP3 (0.56) ACP3TACR1PTPN1PDPK1CNR2
SCHEMBL27664005 0.81 KMT2A (0.51) ACP3TACR1PTPN1PDPK1CNR2
SCHEMBL4433967 0.81 ACP3 (0.41) ACP3TACR1CNR2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP disclosed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed