SCHEMBL4433382

SCHEMBL4433382

COC(=O)c1ccc(-c2ccc3ccccc3c2)[nH]c1=O

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.67
CYP1A2 P05177 1/20 0.67
HPGD P15428 1/20 0.67
HSD17B10 Q99714 1/20 0.67
SLC6A3 Q01959 5/20 0.58
SLC6A2 P23975 4/20 0.58
SLC6A4 P31645 1/20 0.58
PTGER3 P43115 9/20 0.53
KDM4E B2RXH2 3/20 0.50
GAA P10253 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
GLA P06280 1/20 0.50
ALPL P05186 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754413 0.85 PTGER3 (0.56) ALDH1A1CYP1A2HPGDHSD17B10PTGER3
SCHEMBL4431905 0.83 KDM4E (0.69) ALDH1A1CYP1A2HPGDHSD17B10PTGER3
SCHEMBL12427049 0.83 KDM4E (0.64) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3
SCHEMBL4437640 0.83 KDM4E (0.68) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3
SCHEMBL9535126 0.81 PTGER3 (0.54) ALDH1A1CYP1A2HPGDHSD17B10PTGER3
SCHEMBL4431012 0.78 SLC6A3 (0.58) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3
SCHEMBL1547993 0.77 KDM4E (0.55) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3
SCHEMBL4428291 0.76 KDM4E (0.48) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3
SCHEMBL12427050 0.75 CFTR (0.52) ALDH1A1CYP1A2HPGDHSD17B10KDM4E
SCHEMBL9535849 0.75 PTGER3 (0.57) ALDH1A1CYP1A2HPGDHSD17B10SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO claimed
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed