SCHEMBL4431012

SCHEMBL4431012

COC(=O)c1ccc(Cc2ccccc2-c2ccc3ccccc3c2)[nH]c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.58
SLC6A2 P23975 4/20 0.58
SLC6A4 P31645 2/20 0.58
CYP1A2 P05177 4/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 1/20 0.49
HSD17B10 Q99714 1/20 0.49
ALPL P05186 1/20 0.42
KDM4E B2RXH2 2/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
CCNC P24863 2/20 0.40
CDK8 P49336 2/20 0.40
ROCK2 O75116 1/20 0.40
CSF1R P07333 1/20 0.40
KDR P35968 1/20 0.40
FLT3 P36888 1/20 0.40
GSK3A P49840 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438513 0.87 KDM4E (0.47) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1
SCHEMBL4430746 0.86 CYP1A2 (0.48) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1
SCHEMBL4437699 0.85 SLC6A3 (0.55) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1
SCHEMBL4439655 0.82 MAPK8 (0.45) ALDH1A1KDM4EGLAGAAPDE3B
SCHEMBL4428291 0.81 KDM4E (0.48) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1
SCHEMBL4433382 0.78 ALDH1A1 (0.67) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1
SCHEMBL4431808 0.78 KDM4E (0.50) CYP1A2ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL4426834 0.77 ALDH1A1 (0.54) CYP1A2ALDH1A1HSD17B10KDM4EGLA
SCHEMBL4432962 0.75 MDM2 (0.42) ALDH1A1HPGDKDM4EGAAPDE3B
SCHEMBL16683936 0.75 SLC6A3 (1.00) SLC6A3SLC6A2SLC6A4CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed