SCHEMBL4434656

SCHEMBL4434656

COc1cc(F)ccc1CC=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
HPGD P15428 1/20 0.44
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KDM4E B2RXH2 3/20 0.40
APLNR P35414 1/20 0.40
ERN1 O75460 1/20 0.39
NFE2L2 Q16236 1/20 0.39
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29531337 1.00 ALDH1A1 (0.44) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL30536248 0.87 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL2689127 0.87 ALDH1A1 (0.52) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL17423620 0.83 MAPK1 (0.40) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL8436892 0.82 ALDH1A1 (0.47) ALDH1A1POLBHDAC3HDAC1HDAC2
SCHEMBL31299914 0.81 ALDH1A1 (0.44) ALDH1A1HPGDAPLNRERN1GAA
SCHEMBL17537954 0.81 ALDH1A1 (0.50) ALDH1A1KMT2AMEN1KDM4EAPLNR
SCHEMBL17423641 0.81 FFAR4 (0.38) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL8342657 0.81 KDM4E (0.47) ALDH1A1KMT2AMEN1POLBHPGD
SCHEMBL1613798 0.80 APLNR (0.62) ALDH1A1KMT2AMEN1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed