SCHEMBL4435176

SCHEMBL4435176

O=CC(Cl)C1(c2ccccc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
CYP2C9 P11712 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.36
AKR1C1 Q04828 1/20 0.35
HDAC4 P56524 3/20 0.35
OPRM1 P35372 2/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
PNMT P11086 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4445342 0.82 SLC6A4 (0.46) TSHRHDAC4OPRK1MAOAMAOB
SCHEMBL4437272 0.80 LIG1 (0.32) OPRM1OPRK1OPRL1MAOAMAOB
SCHEMBL19207558 0.78 HDAC4 (0.39) MEN1CYP2C9KMT2AAKR1C1HDAC4
SCHEMBL4439597 0.77 SLC6A4 (0.50) TSHRHDAC4OPRK1SLC6A2SLC6A4
SCHEMBL7572201 0.77 SLC6A4 (0.54) TSHRHDAC4OPRK1SLC6A2SLC6A4
SCHEMBL7566171 0.76 SLC6A4 (0.57) TSHRHDAC4OPRK1SLC6A2SLC6A4
SCHEMBL1952823 0.76 SLC6A4 (0.50) MEN1KMT2ATSHROPRM1OPRK1
SCHEMBL4445384 0.75 HDAC4 (0.40) MEN1KMT2ATSHRHDAC4OPRM1
SCHEMBL7563624 0.73 SLC6A4 (0.40) TSHRHDAC4OPRK1SLC6A2SLC6A4
SCHEMBL7571205 0.72 ICMT (0.40) MEN1KMT2ASLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134692-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION Wyeth a Corporation of the State of Delaware (US) 2009-12-23 EP disclosed
WO-2008121817-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION WYETH (US) 2008-10-09 WO disclosed