SCHEMBL4435698

SCHEMBL4435698

Fc1cc(Cl)cc(-c2nc3c(F)cccc3cc2CCNc2ncnc3[nH]cnc23)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.37
LMNA P02545 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
MAPK1 P28482 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.34
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAP4K4 O95819 4/20 0.33
AURKA O14965 2/20 0.33
RPS6KB1 P23443 1/20 0.33
LRRK2 Q5S007 2/20 0.33
STK4 Q13043 1/20 0.33
STK3 Q13188 1/20 0.33
PIK3CD O00329 5/20 0.32
CLK4 Q9HAZ1 2/20 0.32
CDC7 O00311 1/20 0.32
DBF4 Q9UBU7 1/20 0.32
DAPK3 O43293 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16799113 0.94 LMNA (0.39) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4433351 0.89 MAP4K4 (0.41) HTTLMNASMN1; SMN2MAPK1MAP4K4
SCHEMBL4434824 0.87 LMNA (0.42) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4431745 0.86 HTT (0.38) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4434206 0.85 HTT (0.38) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4433726 0.84 HTT (0.37) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4435767 0.84 MAP4K4 (0.40) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4443357 0.84 PIK3CD (0.40) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4433753 0.83 MAPK1 (0.37) HTTLMNASMN1; SMN2MAPK1L3MBTL1
SCHEMBL4443103 0.80 LMNA (0.40) HTTLMNASMN1; SMN2MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137186-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES Amgen Inc. (US) 2009-12-30 EP disclosed
WO-2008118468-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2008-10-02 WO disclosed