SCHEMBL4435833

SCHEMBL4435833

N#Cc1cccc2c1cnn2CCCC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
HSD17B10 Q99714 2/20 0.48
TSHR P16473 1/20 0.48
KMO O15229 6/20 0.47
FABP4 P15090 2/20 0.43
FABP5 Q01469 2/20 0.43
PDE4B Q07343 1/20 0.43
PDE4D Q08499 1/20 0.43
PTGIR P43119 2/20 0.41
FFAR4 Q5NUL3 1/20 0.39
STAT3 P40763 1/20 0.39
HPGD P15428 1/20 0.38
AR P10275 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
SLC22A12 Q96S37 2/20 0.37
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRB1 P18505 1/20 0.37
GABRG2 P18507 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4447530 0.92 KMO (0.56) KDM4EHSD17B10TSHRKMOFABP4
SCHEMBL1398456 0.83 MAPT (0.46) KDM4EHSD17B10PDE4BPDE4D
SCHEMBL13332354 0.80 SLC9A1 (0.41) AR
SCHEMBL13644162 0.80 POLB (0.45) KDM4EHSD17B10TSHRKMOHPGD
SCHEMBL1398508 0.78 MAPT (0.47) KDM4EHSD17B10KMOPDE4BHPGD
SCHEMBL418623 0.76 STAT3 (0.50) TSHRFABP4FABP5STAT3PTGDR2
SCHEMBL22965232 0.74 KMO (0.82) KDM4EHSD17B10TSHRKMOFABP4
SCHEMBL12809063 0.73 CYP1A2 (0.33) AR
SCHEMBL1398518 0.72 MAPT (0.39) KDM4EHSD17B10HPGDAR
SCHEMBL22965217 0.70 KMO (0.51) KDM4EHSD17B10TSHRKMOFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137181-A1 OXADIAZOLE SUBSTITUTED INDAZOLE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE (S1P) AGONISTS Glaxo Group Limited (GB) 2009-12-30 EP disclosed
WO-2008128951-A1 OXADIAZOLE SUBSTITUTED INDAZOLE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE (S1P) AGONISTS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed