SCHEMBL12809063

SCHEMBL12809063

CC1OC(CCCn2ncc3c(C#N)cccc32)O1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
GRM2 Q14416 1/20 0.32
AR P10275 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
IMPDH2 P12268 1/20 0.31
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12600238 0.85
SCHEMBL13332354 0.79 SLC9A1 (0.41) CYP1A2HTR1AADRA1DADRA1AADRA1B
SCHEMBL12600616 0.76 KDM1A (0.33) CYP1A2
SCHEMBL12809065 0.76 ADORA2A (0.31) CYP1A2HTT
SCHEMBL12600620 0.75 HTR2A (0.36) HTT
SCHEMBL12600614 0.74 CYP11B2 (0.37) CYP1A2SLC6A4
SCHEMBL12600913 0.74 KMO (0.30)
SCHEMBL12600921 0.73 CACNA1H (0.34) AR
SCHEMBL15808426 0.72 IMPDH2 (0.43) CYP1A2IMPDH2HTT
SCHEMBL1398456 0.70 MAPT (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137181-B1 OXADIAZOLE SUBSTITUTED INDAZOLE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE (S1P) AGONISTS GLAXO GROUP LTD (GB) 2011-03-02 EP disclosed
WO-2008128951-A1 OXADIAZOLE SUBSTITUTED INDAZOLE DERIVATIVES FOR USE AS SPHINGOSINE 1-PHOSPHATE (S1P) AGONISTS GLAXO GROUP LIMITED (GB) 2008-10-30 WO disclosed