SCHEMBL4436800

SCHEMBL4436800

CN(Cc1ccccc1)[C@@H](CCOC(=O)C(=O)OCC[C@@H](c1cccs1)N(C)Cc1ccccc1)c1cccs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.43
CHRNB4 P30926 2/20 0.43
CHRNA3 P32297 2/20 0.43
CHRNA4 P43681 2/20 0.43
TSHR P16473 2/20 0.42
LMNA P02545 3/20 0.39
TP53 P04637 1/20 0.39
POLB P06746 1/20 0.39
THRB P10828 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4440878 0.82 LMNA (0.41) TSHRLMNATP53POLBTHRB
SCHEMBL4438409 0.82 LMNA (0.41) TSHRLMNATP53POLBTHRB
SCHEMBL4448653 0.82 LMNA (0.41) TSHRLMNATP53POLBTHRB
SCHEMBL11202255 0.79 LMNA (0.43) TSHRLMNATP53POLBTHRB
SCHEMBL15234415 0.71 TSHR (0.50) TSHRLMNATP53POLBTHRB
SCHEMBL6070394 0.70 TSHR (0.42) TSHRLMNATP53POLBTHRB
SCHEMBL13986004 0.68 LMNA (0.43) TSHRLMNACYP3A4CYP2D6ALDH1A1
Oxalic Acid SCHEMBL4436798 0.68 TSHR (0.46) TSHRALDH1A1KDM4EMEN1NPC1
SCHEMBL5914983 0.68 TSHR (0.49) TSHRLMNATP53POLBTHRB
SCHEMBL5914993 0.68 TSHR (0.49) TSHRLMNATP53POLBTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125772-A1 A PROCESS FOR THE PREPARATION OF DULOXETIN AND NEW KEY INTERMEDIATES FOR USE THEREIN Richter Gedeon NYRT (HU) 2009-12-02 EP disclosed
WO-2008078124-A1 A PROCESS FOR THE PREPARATION OF DULOXETIN AND NEW KEY INTERMEDIATES FOR USE THEREIN RICHTER GEDEON NYRT. (HU) 2008-07-03 WO disclosed