SCHEMBL4438532

SCHEMBL4438532

COC(=O)c1ccc(Cc2cccc(-c3ccccc3)c2)[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
GAA P10253 2/20 0.46
GLA P06280 1/20 0.46
MMP1 P03956 2/20 0.44
MMP2 P08253 2/20 0.44
MMP12 P39900 2/20 0.44
PDE10A Q9Y233 1/20 0.44
NR4A2 P43354 2/20 0.43
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
ACLY P53396 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
RNASEH1 O60930 1/20 0.41
MMP9 P14780 1/20 0.41
GPR84 Q9NQS5 1/20 0.41
LIPG Q9Y5X9 1/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4438837 0.90 ALDH1A1 (0.49) ALDH1A1KDM4EGAAGLAPDE3B
SCHEMBL4426842 0.89 KDM4E (0.49) ALDH1A1KDM4EGAAGLANR4A2
SCHEMBL5154097 0.88 KDM4E (0.54) ALDH1A1KDM4EGAAGLAMMP2
SCHEMBL4430692 0.86 KDM4E (0.51) KDM4EMMP1MMP2MMP12ACLY
SCHEMBL4430805 0.84 KDM4E (0.47) ALDH1A1KDM4EGAAGLAMMP1
SCHEMBL4428809 0.84 DAO (0.48) ALDH1A1KDM4EGAAGLAMMP1
SCHEMBL4437957 0.84 PDE3B (0.51) ALDH1A1KDM4EGAAGLAMMP1
SCHEMBL4428291 0.82 KDM4E (0.48) ALDH1A1KDM4EGAAGLAPDE10A
SCHEMBL4426834 0.81 ALDH1A1 (0.54) ALDH1A1KDM4EGAAGLAPDE3B
SCHEMBL4429436 0.79 KDM4E (0.53) ALDH1A1KDM4EGAAGLAMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed