SCHEMBL4438837

SCHEMBL4438837

COC(=O)c1ccc(Cc2cccc(Cc3ccccc3)c2)[nH]c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
KDM4E B2RXH2 4/20 0.49
GAA P10253 2/20 0.48
GLA P06280 1/20 0.48
RNASEH1 O60930 1/20 0.45
TSHR P16473 3/20 0.44
MAPT P10636 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
NFKB1 P19838 1/20 0.44
CYP2C19 P33261 1/20 0.44
BLM P54132 1/20 0.44
PMP22 Q01453 1/20 0.44
HIF1A Q16665 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HSD17B10 Q99714 3/20 0.43
HPGD P15428 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5154097 0.93 KDM4E (0.54) ALDH1A1KDM4EGAAGLARNASEH1
SCHEMBL4438532 0.90 ALDH1A1 (0.47) ALDH1A1KDM4EGAAGLARNASEH1
SCHEMBL4428809 0.86 DAO (0.48) ALDH1A1KDM4EGAAGLAMAPT
SCHEMBL4437957 0.86 PDE3B (0.51) ALDH1A1KDM4EGAAGLAMAPT
SCHEMBL4430805 0.86 KDM4E (0.47) ALDH1A1KDM4EGAAGLATSHR
SCHEMBL4426834 0.86 ALDH1A1 (0.54) ALDH1A1KDM4EGAAGLARNASEH1
SCHEMBL4426842 0.86 KDM4E (0.49) ALDH1A1KDM4EGAAGLARNASEH1
SCHEMBL4432424 0.85 HNF4A (0.49) KDM4ERNASEH1PARP1MPODAO
SCHEMBL4428291 0.85 KDM4E (0.48) ALDH1A1KDM4EGAAGLARNASEH1
SCHEMBL4429436 0.81 KDM4E (0.53) ALDH1A1KDM4EGAAGLARNASEH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125739-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2009-12-02 EP disclosed
WO-2008079371-A1 MODULATORS OF C3A RECEPTOR AND METHODS OF USE THEREOF ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-07-03 WO disclosed