SCHEMBL4440422

SCHEMBL4440422

O=CCC(c1ccc(C(F)(F)F)cc1)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 3/20 0.43
TRPM8 Q7Z2W7 1/20 0.39
FFAR1 O14842 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
CTSA P10619 1/20 0.38
GPR139 Q6DWJ6 1/20 0.37
ACP3 P15309 1/20 0.37
KIF11 P52732 1/20 0.36
CACNA1A O00555 2/20 0.36
CACNA2D1 P54289 2/20 0.36
CACNB1 Q02641 2/20 0.36
CACNA1C Q13936 2/20 0.36
CACNA1B Q00975 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4434672 0.89 PPARG (0.41) FFAR1ACP3CACNA1ACACNA2D1CACNB1
SCHEMBL6703510 0.82 ACP3 (0.51) ACP3KIF11CACNA1ACACNA2D1CACNB1
SCHEMBL4433877 0.80 ACP3 (0.39) FFAR1ACP3CACNA1ACACNA2D1CACNB1
SCHEMBL4441831 0.80 CASR (0.35) MMP2MMP9ACP3CACNA1ACACNA2D1
SCHEMBL23960436 0.74 CYP19A1 (0.46) FFAR1ACP3CACNA1ACACNA2D1CACNB1
SCHEMBL4441719 0.74 AKR1C3 (0.46)
SCHEMBL25954028 0.72 CHRM2 (0.41) CETPCHRM2CHRM1CHRM3GPR139
SCHEMBL4970158 0.70 GPR139 (0.50) CETPTRPM8CTSAGPR139
SCHEMBL22089163 0.69 CTSA (0.53) TRPM8FFAR1CTSA
SCHEMBL25336167 0.69 CHRM2 (0.39) CETPCHRM2CHRM1CHRM3GPR139

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed