SCHEMBL4434672

SCHEMBL4434672

O=CCC(c1ccc(C(F)(F)F)cc1)c1cccc(OC(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.41
PPARA Q07869 2/20 0.41
FFAR1 O14842 3/20 0.40
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DRD1 P21728 1/20 0.39
CACNA1C Q13936 2/20 0.38
CACNA1A O00555 2/20 0.38
CACNA2D1 P54289 2/20 0.38
CACNB1 Q02641 2/20 0.38
CACNA1B Q00975 1/20 0.38
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
SLC6A3 Q01959 2/20 0.38
KCNK2 O95069 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4440422 0.89 CETP (0.43) FFAR1CACNA1CCACNA1ACACNA2D1CACNB1
SCHEMBL6703510 0.81 ACP3 (0.51) CACNA1CCACNA1ACACNA2D1CACNB1CACNA1B
SCHEMBL4433877 0.79 ACP3 (0.39) PPARGFFAR1CACNA1CCACNA1ACACNA2D1
SCHEMBL4431369 0.74 MEN1 (0.43) PPARGPPARAFFAR1MEN1LMNA
SCHEMBL22965330 0.74 DRD1 (0.46) MEN1LMNAMAPTHTTKMT2A
SCHEMBL23960436 0.73 CYP19A1 (0.46) FFAR1CACNA1CCACNA1ACACNA2D1CACNB1
SCHEMBL4441719 0.73 AKR1C3 (0.46) PPARGPPARAMEN1KMT2A
SCHEMBL4435507 0.72 KDM4E (0.45) MEN1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL4431243 0.72 KDM4E (0.45) MEN1LMNAHTTKMT2ASMN1; SMN2
SCHEMBL4431325 0.72 KDM4E (0.45) MEN1LMNAHTTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed