SCHEMBL4433877

SCHEMBL4433877

O=CCC(c1ccc(C(F)(F)F)cc1)c1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 2/20 0.39
CASR P41180 2/20 0.39
FFAR2 O15552 1/20 0.39
GRIN2B Q13224 1/20 0.39
CACNA1A O00555 1/20 0.38
CACNA2D1 P54289 1/20 0.38
CACNA1B Q00975 1/20 0.38
CACNB1 Q02641 1/20 0.38
CACNA1C Q13936 1/20 0.38
GAA P10253 1/20 0.38
PPARG P37231 3/20 0.38
TACR1 P25103 2/20 0.37
OPRL1 P41146 1/20 0.36
FFAR1 O14842 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6703510 0.85 ACP3 (0.51) ACP3CACNA1ACACNA2D1CACNA1BCACNB1
SCHEMBL6699162 0.85 ACP3 (0.47) ACP3CASRCACNA2D1CACNA1BCACNB1
SCHEMBL1581317 0.81 PNMT (0.45) ACP3CASRFFAR2GRIN2BCACNA1C
SCHEMBL4440422 0.80 CETP (0.43) ACP3CACNA1ACACNA2D1CACNA1BCACNB1
SCHEMBL4434672 0.79 PPARG (0.41) ACP3CACNA1ACACNA2D1CACNA1BCACNB1
SCHEMBL23960436 0.77 CYP19A1 (0.46) ACP3CACNA1ACACNA2D1CACNA1BCACNB1
SCHEMBL27614458 0.77 LMNA (0.36) ACP3CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL6339476 0.75 PPARG (0.39) PPARGOPRL1CNR1CNR2
SCHEMBL4441831 0.75 CASR (0.35) ACP3CASRCACNA1ACACNA2D1CACNA1B
SCHEMBL4441719 0.74 AKR1C3 (0.46) CASRPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114867-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. Hoffmann-Roche AG (CH) 2009-11-11 EP disclosed
WO-2008107335-A1 AMINOAMIDES AS OREXIN ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2008-09-12 WO disclosed