SCHEMBL4440443

SCHEMBL4440443

CCOC(=O)c1ccc(CNC(C)NCc2ccc(C(=O)OCC)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.63
HTT P42858 3/20 0.57
MAPT P10636 3/20 0.55
L3MBTL1 Q9Y468 3/20 0.55
RAB9A P51151 2/20 0.55
ALDH1A1 P00352 2/20 0.55
NPC1 O15118 1/20 0.55
CA1 P00915 2/20 0.54
CA2 P00918 2/20 0.54
CA12 O43570 1/20 0.54
ESR1 P03372 1/20 0.54
CA7 P43166 1/20 0.54
CA9 Q16790 1/20 0.54
ESR2 Q92731 1/20 0.54
CA14 Q9ULX7 1/20 0.54
LMNA P02545 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
MAOA P21397 1/20 0.53
KMT2A Q03164 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4430709 0.85 LOXL2 (0.58) SMN1; SMN2MAPTRAB9ANPC1CA1
SCHEMBL2145311 0.83 SMN1; SMN2 (0.58) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL11988605 0.81 SMN1; SMN2 (0.69) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL4712796 0.81 SMN1; SMN2 (0.68) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL7746905 0.80 CA1 (0.79) SMN1; SMN2HTTMAPTRAB9AALDH1A1
SCHEMBL25232330 0.80 SMN1; SMN2 (0.77) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL7322209 0.80 HTT (0.73) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL2940862 0.80 SMN1; SMN2 (0.77) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL28120177 0.80 SMN1; SMN2 (0.67) SMN1; SMN2HTTMAPTL3MBTL1RAB9A
SCHEMBL9125949 0.79 HTT (0.67) SMN1; SMN2HTTMAPTL3MBTL1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114899-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES Firmenich S.A. (CH) 2009-11-11 EP claimed
WO-2008093272-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES FIRMENICH SA (CH) 2008-08-07 WO claimed
EP-2114899-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES Firmenich S.A. (CH) 2009-11-11 EP disclosed
WO-2008093272-A2 CONTROLLED RELEASE OF ACTIVE ALDEHYDES AND KETONES FROM EQUILIBRATED DYNAMIC MIXTURES FIRMENICH SA (CH) 2008-08-07 WO disclosed