SCHEMBL4440469

SCHEMBL4440469

O=CC(O)C1(c2ccc(OC(F)(F)F)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.50
SLC6A3 Q01959 9/20 0.50
SLC6A2 P23975 2/20 0.50
NR1I2 O75469 1/20 0.44
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
EPHX2 P34913 1/20 0.38
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4446504 0.80 MAOA (0.39) SLC6A4SLC6A3SLC6A2PIM1PIM2
SCHEMBL4436040 0.77 HSD11B1 (0.37) SLC6A3KMT2A
SCHEMBL4283467 0.77 SLC6A4 (0.55) SLC6A4SLC6A3SLC6A2NR1I2PIM1
SCHEMBL20886289 0.77 SLC6A4 (0.55) SLC6A4SLC6A3SLC6A2NR1I2PIM1
SCHEMBL10157208 0.76 SLC6A4 (0.65) SLC6A4SLC6A3SLC6A2NR1I2
SCHEMBL4438204 0.74 CYP2A6 (0.34) SLC6A3KMT2A
SCHEMBL8535883 0.72 SLC6A4 (0.45) SLC6A4SLC6A3SLC6A2PIM1PIM2
SCHEMBL4554666 0.71 SLC6A4 (0.44) SLC6A4SLC6A3SLC6A2PIM1PIM2
SCHEMBL625374 0.70 SLC6A4 (0.47) SLC6A4SLC6A3SLC6A2PIM1PIM2
SCHEMBL19955250 0.69 SLC6A4 (0.43) SLC6A4SLC6A3SLC6A2PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2134692-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION Wyeth a Corporation of the State of Delaware (US) 2009-12-23 EP disclosed
WO-2008121817-A2 QUINOLINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM FOR SELECTIN INHIBITION WYETH (US) 2008-10-09 WO disclosed