SCHEMBL4442452

SCHEMBL4442452

OB(O)c1cc2cc(CCCc3ccccc3)ccc2o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
MGLL Q99685 1/20 0.54
HSD17B10 Q99714 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
FFAR1 O14842 1/20 0.44
IGF1R P08069 1/20 0.41
ALOX15 P16050 1/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA3 P07451 1/20 0.40
CA4 P22748 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
S1PR1 P21453 1/20 0.40
HTR2A P28223 1/20 0.39
CYP1A2 P05177 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442995 0.94 KDM4E (0.57) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL1601545 0.85 KDM4E (0.57) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL1602662 0.84 MGLL (0.47) KDM4EMGLLHSD17B10TDP1CA1
SCHEMBL1603585 0.77 KDM4E (0.51) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL1602396 0.77 KDM4E (0.46) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL1602638 0.75 KDM4E (0.49) KDM4EMGLLHSD17B10TDP1S1PR1
SCHEMBL14677067 0.75 ALDH1A1 (0.52) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL7463907 0.74 LPL (0.49) KDM4EMGLLHSD17B10TDP1CA1
SCHEMBL1600996 0.73 KDM4E (0.50) KDM4EMGLLHSD17B10TDP1FFAR1
SCHEMBL1601191 0.73 KDM4E (0.62) KDM4EMGLLHSD17B10TDP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121648-A2 S1P RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
WO-2007109334-A2 SIP RECEPTOR MODULATING COMPOUNDS AND USE THEREOF EPIX DELAWARE, INC. (US) 2007-09-27 WO disclosed