SCHEMBL444400

SCHEMBL444400

[CH]1C=NOc2ccccc21

nearest known ligand 0.34

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8480733 0.76 KDM4E (0.36) TRPA1
SCHEMBL29757278 0.76 KDM4E (0.36) TRPA1
Urea SCHEMBL8887498 0.69 KDM4E (0.35) TRPA1
Oxalic Acid SCHEMBL10499933 0.69 MEN1 (0.32)
Acetic Acid SCHEMBL25341096 0.68 TRPA1 (0.31) TRPA1
Fumaric Acid SCHEMBL11602682 0.66 ALDH1A1 (0.38)
SCHEMBL218834 0.64 TRPA1 (0.36) TRPA1
SCHEMBL6118600 0.63
SCHEMBL23400 0.62 KDM4E (0.35) TRPA1
SCHEMBL209689 0.62 TRPA1 (0.34) TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 483 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3642202-A1 DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES Pfizer Inc (US) 2020-04-29 EP claimed
EP-3478679-A1 5,7-DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES FOR TREATING NEUROLOGICAL AND NEURODEGENERATIVE DISEASES Pfizer Inc (US) 2019-05-08 EP claimed
EP-3419979-A1 6,7-DIHYDRO-5H-PYRAZOLO[5,1-B][1,3]OXAZINE-2-CARBOXAMIDE COMPOUNDS Pfizer Inc (US) 2019-01-02 EP claimed
WO-2018234953-A1 DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES PFIZER INC. (US) 2018-12-27 WO claimed
EP-3310784-A1 TRICYCLIC COMPOUNDS AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS Pfizer Inc (US) 2018-04-25 EP claimed
WO-2018002760-A1 5,7-DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES FOR TREATING NEUROLOGICAL AND NEURODEGENERATIVE DISEASES PFIZER INC. (US) 2018-01-04 WO claimed
WO-2017145013-A1 6,7-DIHYDRO-5H-PYRAZOLO[5,1-B][1,3]OXAZINE-2-CARBOXAMIDE COMPOUNDS PFIZER INC. (US) 2017-08-31 WO claimed
EP-3177624-A1 IMIDAZOPYRIDAZINE COMPOUNDS Pfizer Inc (US) 2017-06-14 EP claimed
WO-2016203347-A1 TRICYCLIC COMPOUNDS AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS PFIZER INC. (US) 2016-12-22 WO claimed
WO-2016020786-A1 IMIDAZOPYRIDAZINE COMPOUNDS PFIZER INC. (US) 2016-02-11 WO claimed
CN-1074413-C Novel benzimidazole derivatives having CGMP-phosphodisterase inhibiting activity OTSUKA PHARMA CO LTD (JP) 2001-11-07 CN claimed
CN-1070856-C Thiazole derivatives OTSUDA PHARMACEUTICAL CO LTD (JP) 2001-09-12 CN claimed
CN-1275123-A Prostaglandin agonists and their use to treat bone disorders PFIZER (US) 2000-11-29 CN claimed
EP-0570006-B1 A silver halide photographic light-sensitive material FUJI PHOTO FILM CO LTD (JP) 1999-03-24 EP claimed
CN-1198160-A Thiazole derivative OTSUKA PHARMA CO LTD (JP) 1998-11-04 CN claimed
EP-0858452-A1 THIAZOLE DERIVATIVE AS PROTEIN KINASE C INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-08-19 EP claimed
WO-1998004536-A1 THIAZOLE DERIVATIVE AS PROTEIN KINASE C INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1998-02-05 WO claimed
CN-1158129-A Novel benzimidazole derivatives having CGMP-phosphodisterase inhibiting activity OTSUKA PHARMA CO LTD (JP) 1997-08-27 CN claimed
US-5362617-A Multilayer element of support with color couplers FUJI PHOTO FILM CO., LTD. (JP) 1994-11-08 US claimed
EP-0570006-A1 A silver halide photographic light-sensitive material FUJI PHOTO FILM CO., LTD. (JP) 1993-11-18 EP claimed