Temozolomide

Temozolomide

SCHEMBL4444959

Cn1nnc2c(C(N)=O)ncn2c1=O.S=P(N1CC1)(N1CC1)N1CC1

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.78
PABPC1 P11940 1/20 0.78
KMT2A Q03164 1/20 0.78
CA12 O43570 3/20 0.46
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA9 Q16790 3/20 0.46
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Temozolomide SCHEMBL3270220 0.88 MEN1 (1.00) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL3739 0.88 MEN1 (1.00) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL28275477 0.87 MEN1 (0.97) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL3784250 0.87 MEN1 (0.97) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL4746638 0.87 MEN1 (0.97) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL1534013 0.87 MEN1 (0.97) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL27721442 0.86 MEN1 (0.89) MEN1PABPC1KMT2ACA12CA1
SCHEMBL892333 0.80 MEN1 (0.78) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL16227379 0.80 MEN1 (0.82) MEN1PABPC1KMT2ACA12CA1
Temozolomide SCHEMBL10168201 0.79 MEN1 (0.81) MEN1PABPC1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3982977-A1 METHODS OF TREATING CANCER WITH AN INHIBITOR OF ZNF827 Children's Medical Research Institute (AU) 2022-04-20 EP disclosed
WO-2020248018-A1 METHODS OF TREATING CANCER WITH AN INHIBITOR OF ZNF827 CHILDREN'S MEDICAL RESEARCH INSTITUTE (AU) 2020-12-17 WO disclosed
US-10669260-B2 Compounds targeting proteins, compositions, methods, and uses thereof BIOTHERYX, INC. (US) 2020-06-02 US disclosed
CN-110461315-A Treatment and Prevention of Cytokine Release Syndrome Using Chimeric Antigen Receptors in Combination with Kinase Inhibitors NOVARTIS AG 2019-11-15 CN disclosed
CN-108700590-A Cell population analysis 英国质谱公司 2018-10-23 CN disclosed
US-20180065952-A1 COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. 2018-03-08 US disclosed
CN-107667288-A Spectral analysis of microorganisms 英国质谱公司 2018-02-06 CN disclosed
EP-2131840-A1 COMBINATION OF BENZIMIDAZOLE ANTI-CANCER AGENT AND A SECOND ANTI-CANCER AGENT S*Bio Pte Ltd (SG) 2009-12-16 EP disclosed
WO-2008108741-A1 COMBINATION OF BENZIMIDAZOLE ANTI-CANCER AGENT AND A SECOND ANTI-CANCER AGENT S*BIO PTE LTD (SG) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180065952-A1 COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF IKZF3, IKZF1, APC MEN1 3927/4885PABPC1 2075/4885KMT2A 4004/4885
US-10669260-B2 Compounds targeting proteins, compositions, methods, and uses thereof IKZF3, IKZF1, APC MEN1 3927/4885PABPC1 2075/4885KMT2A 4004/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.