SCHEMBL4445468

SCHEMBL4445468

CN(C)S(=O)(=O)ON1CCN(C[C@@H]2OC(=O)N(c3ccc(C(F)(F)F)cc3)[C@H]2c2cccc(F)c2)CC1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.34
KMT2A Q03164 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31
CYP3A4 P08684 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA9 Q16790 1/20 0.31
CCR5 P51681 4/20 0.31
PLD2 O14939 1/20 0.30
PLD1 Q13393 1/20 0.30
KCNH2 Q12809 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13168227 0.88 LMNA (0.34) KMT2ACYP3A4CA1CA2CA9
SCHEMBL3595014 0.86 NTRK1 (0.32) CYP3A4CA1CA2CA9CCR5
SCHEMBL3592352 0.83 ALDH1A1 (0.36) KMT2ADRD2HTR7CCR5KCNH2
SCHEMBL3591176 0.74 KCNN4 (0.36) KCNN4
SCHEMBL3599584 0.73 MAPK14 (0.37) KMT2A
Sulfamide SCHEMBL4438457 0.73 CA1 (0.35) KMT2AHTR2ANR1H2NR1H3CA1
SCHEMBL4441032 0.72 DRD2 (0.41) KMT2ADRD2HTR7CYP3A4
SCHEMBL3595202 0.72 KMT2A (0.38) KMT2AHTR1ADRD2HTR2AHTR7
SCHEMBL4439801 0.72 KMT2A (0.38) KMT2AHTR1ADRD2HTR2AHTR7
SCHEMBL3589557 0.72 GRM5 (0.40) KCNN4KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121598-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2009-11-25 EP claimed
WO-2008076754-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2008-06-26 WO claimed