SCHEMBL4447381

SCHEMBL4447381

CCC(C(=O)C(C(=O)CF)C(N)C(=O)OC(C)(C)C)c1ccnn(Cc2cccc(OC)c2)c1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.37
ALDH1A1 P00352 3/20 0.37
GAA P10253 1/20 0.37
NPBWR1 P48145 2/20 0.35
FPR1 P21462 1/20 0.34
FPR3 P25089 1/20 0.34
FPR2 P25090 1/20 0.34
SLC16A3 O15427 1/20 0.34
SLC16A1 P53985 1/20 0.34
MCTS1 Q9ULC4 1/20 0.34
AURKA O14965 2/20 0.34
GRK2 P25098 1/20 0.34
ROCK1 Q13464 1/20 0.34
RPS6KA1 Q15418 1/20 0.34
ROCK2 O75116 2/20 0.34
PPARG P37231 2/20 0.33
PPARA Q07869 2/20 0.33
PPARD Q03181 1/20 0.33
HCAR3 P49019 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4256061 0.91 NPSR1 (0.38) ALDH1A1NPBWR1KDM4EHSD17B10
SCHEMBL4451133 0.90 PKM (0.42) PKMALDH1A1GAANPBWR1FPR1
SCHEMBL4253173 0.82 NPBWR1 (0.34) ALDH1A1GAANPBWR1KDM4E
SCHEMBL4253283 0.79 CACNA1B (0.38) PKMALDH1A1GAANPBWR1FPR1
SCHEMBL4257924 0.79 HTT (0.41) PKMALDH1A1NPBWR1KDM4E
SCHEMBL4253284 0.77 FPR1 (0.38) PKMALDH1A1GAAFPR1FPR3
SCHEMBL4255683 0.77 PKM (0.47) PKMALDH1A1GAANPBWR1FPR1
SCHEMBL4447384 0.74 PKM (0.37) PKMALDH1A1GAANPBWR1FPR1
SCHEMBL4257238 0.74 PKM (0.41) PKMALDH1A1GAAFPR1FPR3
SCHEMBL13608163 0.74 PKM (0.41) PKMALDH1A1GAAFPR1FPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8481537-B2 Caspase inhibitors based of pyridazinone scaffold LG LIFE SCIENCES LTD. (KR) 2013-07-09 US disclosed
EP-2046757-A1 CASPASE INHIBITORS BASED ON PYRIDAZINONE SCAFFOLD LG Life Sciences Ltd. (KR) 2009-04-15 EP disclosed
WO-2008016239-A1 CASPASE INHIBITORS BASED ON PYRIDAZINONE SCAFFOLD LG LIFE SCIENCES LTD. (KR) 2008-02-07 WO disclosed