SCHEMBL4447829

SCHEMBL4447829

C=CCOCC(C)(C)NC(=O)O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12974868 0.81 SMN1; SMN2 (0.38) TDP1
SCHEMBL2870617 0.80 TDP1 (0.30) TDP1
SCHEMBL30687350 0.76 MGAM (0.36) ALDH1A1
SCHEMBL12581238 0.76 ACLY (0.35) ALDH1A1CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL6279972 0.75
SCHEMBL21340475 0.75 TSHR (0.38) CYP2C19TDP1
SCHEMBL20547591 0.75 PIK3CD (0.31)
SCHEMBL233302 0.74 KMT2A (0.38) ALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL4612722 0.73
SCHEMBL3507606 0.73 TSHR (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11390604-B2 Imidazole-pyrazole derivatives HOFFMANN-LA ROCHE INC. (US) 2022-07-19 US disclosed
EP-3934756-A1 NOVEL IMIDAZOLE-PYRAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2022-01-12 EP disclosed
WO-2020182648-A1 NOVEL IMIDAZOLE-PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2020-09-17 WO disclosed
US-20200290998-A1 NOVEL IMIDAZOLE-PYRAZOLE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2020-09-17 US disclosed
EP-2120965-B1 N-HALOGENATED AMINO COMPOUNDS AND DERIVATIVES NOVABAY PHARMACEUTICALS INC (US) 2014-11-05 EP disclosed
EP-2120965-A1 N-HALOGENATED AMINO COMPOUNDS AND DERIVATIVES Novabay Pharmaceuticals, Inc. (US) 2009-11-25 EP disclosed
WO-2008083347-A1 N-HALOGENATED AMINO COMPOUNDS AND DERIVATIVES NOVABAY PHARMACEUTICALS, INC. (US) 2008-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200290998-A1 NOVEL IMIDAZOLE-PYRAZOLE DERIVATIVES F12, RIN1, CYP3A7 ALDH1A1 951/4885CYP3A4 10/4885CYP2C9 35/4885
US-11390604-B2 Imidazole-pyrazole derivatives F12, CYP3A7, NLRP3 ALDH1A1 912/4885CYP3A4 10/4885CYP2C9 27/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.